SCHEMBL20002927

SCHEMBL20002927

Cc1cc(S(=O)(=O)C2CCN(C(=O)C3CCCCC3)C2)ccc1F

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
CNR1 P21554 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
RORC P51449 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.42
GAA P10253 1/20 0.42
NPC1 O15118 1/20 0.41
GFER P55789 1/20 0.41
HSD11B1 P28845 1/20 0.41
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002703 0.91 ALDH1A1 (0.46) ALDH1A1CNR1NPSR1RORCL3MBTL1
SCHEMBL20003061 0.90 RORC (0.54) RORC
SCHEMBL20002434 0.83 L3MBTL1 (0.56) ALDH1A1NPSR1RORCL3MBTL1HSD11B1
SCHEMBL20002381 0.83 L3MBTL1 (0.56) ALDH1A1NPSR1RORCL3MBTL1HSD11B1
SCHEMBL20002920 0.79 ALDH1A1 (0.46) ALDH1A1CNR1NPSR1L3MBTL1NPC1
SCHEMBL20003180 0.78 RORC (0.54) RORC
SCHEMBL20002822 0.77 RORC (0.58) RORC
SCHEMBL20002251 0.74 RORC (0.52) ALDH1A1RORCL3MBTL1
SCHEMBL20002731 0.74 L3MBTL1 (0.48) ALDH1A1RORCL3MBTL1GAA
SCHEMBL20002254 0.74 L3MBTL1 (0.48) ALDH1A1RORCL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed