SCHEMBL20002953

SCHEMBL20002953

CC(C)(C(=O)N1CCC(S(=O)(=O)c2ccc(F)cc2)C1)n1cccn1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.53
HTR2A P28223 5/20 0.40
HTR2C P28335 4/20 0.40
KCNH2 Q12809 4/20 0.40
EPHX2 P34913 1/20 0.39
DRD2 P14416 2/20 0.37
NAMPT P43490 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
GPR6 P46095 1/20 0.36
MMP13 P45452 1/20 0.36
ALOX5 P09917 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
GCK P35557 1/20 0.35
JAK1 P23458 2/20 0.35
JAK2 O60674 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002244 0.81 RORC (0.46) RORCHTR2AHTR2CKCNH2EPHX2
SCHEMBL20002210 0.78 RORC (0.44) RORCDRD2JAK1JAK2
SCHEMBL20002448 0.78 EPHX2 (0.44) RORCHTR2AHTR2CKCNH2EPHX2
SCHEMBL21426003 0.77 MMP13 (0.53) RORCNAMPTMMP13
SCHEMBL21426007 0.77 MMP13 (0.53) RORCNAMPTMMP13
SCHEMBL14413535 0.73 EPHX2 (0.47) RORCHTR2AHTR2CKCNH2EPHX2
SCHEMBL20003003 0.73 EPHX2 (0.45) RORCHTR2AHTR2CKCNH2EPHX2
SCHEMBL13890294 0.73 EPHX2 (0.50) HTR2AHTR2CKCNH2EPHX2DRD2
SCHEMBL20002502 0.72 L3MBTL1 (0.64) NAMPTMMP13L3MBTL1
SCHEMBL4777810 0.72 MMP13 (0.58) RORCNAMPTMMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed