SCHEMBL20002502

SCHEMBL20002502

O=C(c1cccnc1)N1CCC(S(=O)(=O)c2ccc(F)cc2)C1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.64
SLC18A3 Q16572 2/20 0.56
RAB9A P51151 1/20 0.53
ALDH1A1 P00352 3/20 0.52
LMNA P02545 1/20 0.49
PTGS2 P35354 1/20 0.49
MAPK1 P28482 1/20 0.49
POLB P06746 1/20 0.48
CHRNB2 P17787 1/20 0.47
CHRNB4 P30926 1/20 0.47
CHRNA3 P32297 1/20 0.47
CHRNA7 P36544 1/20 0.47
CHRNA4 P43681 1/20 0.47
NAMPT P43490 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
GAA P10253 1/20 0.47
MMP1 P03956 1/20 0.46
MMP3 P08254 1/20 0.46
MMP7 P09237 1/20 0.46
MMP9 P14780 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003002 0.83 TSHR (0.48) L3MBTL1RAB9AALDH1A1MAPK1NAMPT
SCHEMBL20003085 0.81 PROKR1 (0.44) L3MBTL1RAB9APOLBNAMPTGAA
SCHEMBL20003091 0.80 RORC (0.54) L3MBTL1RAB9AALDH1A1LMNANAMPT
SCHEMBL20002270 0.77 KMT2A (0.60) RAB9AALDH1A1LMNASMN1; SMN2
SCHEMBL14413535 0.76 EPHX2 (0.47) L3MBTL1POLBCYP3A4
SCHEMBL20003016 0.76 RORC (0.50) L3MBTL1RAB9AALDH1A1LMNAPOLB
SCHEMBL6209453 0.76 SLC18A3 (0.75) SLC18A3POLBGAA
SCHEMBL20003147 0.76 RORC (0.51) RAB9AALDH1A1
SCHEMBL20002837 0.75 RORC (0.49) ALDH1A1NAMPTSMN1; SMN2
SCHEMBL15017250 0.75 VNN1 (0.65) SLC18A3ALDH1A1MAPK1POLBCHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed