SCHEMBL20002976

SCHEMBL20002976

Cc1cc([S+]([O-])C2CCN(C(=O)C34CCC(C(=O)O)(CC3)CC4)C2)ccc1F

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RORC P51449 15/20 0.43
DRD4 P21917 2/20 0.33
HSD11B1 P28845 2/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002767 0.92 RORC (0.43) RORCHSD11B1
SCHEMBL20003077 0.88 RORC (0.48) RORCDRD4HCRTR1HCRTR2
SCHEMBL20003044 0.85 RORC (0.40) RORC
SCHEMBL20002735 0.83 RORC (0.47) RORC
SCHEMBL20002561 0.82 RORC (0.50) RORC
SCHEMBL20003094 0.80 TACR3 (0.33) RORCDRD4HCRTR1HCRTR2
SCHEMBL20003010 0.79 RORC (0.43) RORC
SCHEMBL20003110 0.79 RORC (0.41) RORCDRD4HCRTR1HCRTR2
SCHEMBL20003241 0.79 RORC (0.41) RORCHSD11B1
SCHEMBL20003180 0.76 RORC (0.54) RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed