SCHEMBL20003094

SCHEMBL20003094

CCOC1(C(=O)N2CCC([S+]([O-])c3ccc(F)c(C)c3)C2)CCC(C)(C(=O)O)CC1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 2/20 0.33
RORC P51449 4/20 0.33
GRIN2B Q13224 2/20 0.32
RECQL P46063 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
KDM4E B2RXH2 2/20 0.31
HSD17B10 Q99714 1/20 0.31
ALDH1A1 P00352 3/20 0.31
SMN1; SMN2 Q16637 3/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
DRD4 P21917 1/20 0.31
MGLL Q99685 1/20 0.30
EPHX2 P34913 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002976 0.80 RORC (0.43) RORCHCRTR1HCRTR2DRD4
SCHEMBL20002561 0.80 RORC (0.50) RORCGRIN2B
SCHEMBL20003110 0.79 RORC (0.41) RORCGRIN2BHCRTR1HCRTR2DRD4
SCHEMBL20002735 0.76 RORC (0.47) RORC
SCHEMBL20003077 0.75 RORC (0.48) RORCHCRTR1HCRTR2DRD4
SCHEMBL20002767 0.72 RORC (0.43) RORCSMN1; SMN2LMNA
SCHEMBL20003010 0.72 RORC (0.43) RORCALDH1A1
SCHEMBL20002748 0.67 RORC (0.39) RORCALDH1A1SMN1; SMN2KMT2ALMNA
SCHEMBL20002622 0.66 RORC (0.49) RORCALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL20003044 0.66 RORC (0.40) RORCALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed