SCHEMBL20003016

SCHEMBL20003016

O=C(c1ccc(=O)[nH]c1)N1CCC(S(=O)(=O)c2ccc(F)cc2)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.50
HTR2A P28223 2/20 0.44
HTR2C P28335 1/20 0.44
KCNH2 Q12809 1/20 0.44
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ATM Q13315 1/20 0.43
TRPV6 Q9H1D0 1/20 0.43
CYP2C9 P11712 1/20 0.42
SLC9A1 P19634 1/20 0.42
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003147 0.79 RORC (0.51) RORCHTR2AHTR2CKCNH2CA12
SCHEMBL20002270 0.79 KMT2A (0.60) HTR2AHTR2CKCNH2CA12CA1
SCHEMBL20002502 0.76 L3MBTL1 (0.64) RAB9AALDH1A1L3MBTL1LMNAPOLB
SCHEMBL14413535 0.76 EPHX2 (0.47) RORCHTR2AHTR2CKCNH2CA12
SCHEMBL20003085 0.76 PROKR1 (0.44) HTR2AHTR2CKCNH2CA12CA1
SCHEMBL20003003 0.75 EPHX2 (0.45) RORCHTR2AHTR2CKCNH2CA12
SCHEMBL13890294 0.72 EPHX2 (0.50) HTR2AHTR2CKCNH2NPC1RAB9A
SCHEMBL20002563 0.72 EPHX2 (0.45) HTR2AHTR2CKCNH2ALDH1A1KDM4E
SCHEMBL20003057 0.72 RORC (0.50) RORCHTR2AHTR2CKCNH2CA12
SCHEMBL20002381 0.72 L3MBTL1 (0.56) RORCCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed