SCHEMBL20003085

SCHEMBL20003085

O=C(c1ccnc(O)c1)N1CCC(S(=O)(=O)c2ccc(F)cc2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 1/20 0.44
NAMPT P43490 5/20 0.44
EPHX2 P34913 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
KCNH2 Q12809 1/20 0.42
HSD11B1 P28845 4/20 0.41
AKT1 P31749 1/20 0.41
PIK3CA P42336 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ATM Q13315 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002502 0.81 L3MBTL1 (0.64) NAMPTL3MBTL1RAB9APOLBGAA
SCHEMBL20002270 0.76 KMT2A (0.60) HTR2AHTR2CKCNH2HSD11B1CA12
SCHEMBL14413535 0.76 EPHX2 (0.47) EPHX2HTR2AHTR2CKCNH2L3MBTL1
SCHEMBL20003016 0.76 RORC (0.50) NAMPTEPHX2HTR2AHTR2CKCNH2
SCHEMBL20003147 0.75 RORC (0.51) EPHX2HTR2AHTR2CKCNH2HSD11B1
SCHEMBL20003003 0.72 EPHX2 (0.45) EPHX2HTR2AHTR2CKCNH2L3MBTL1
SCHEMBL20002563 0.72 EPHX2 (0.45) EPHX2HTR2AHTR2CKCNH2L3MBTL1
SCHEMBL13890294 0.72 EPHX2 (0.50) EPHX2HTR2AHTR2CKCNH2L3MBTL1
SCHEMBL20002837 0.72 RORC (0.49) NAMPTEPHX2HTR2AHTR2CKCNH2
SCHEMBL20003031 0.72 EPHX2 (0.44) NAMPTEPHX2HTR2AHTR2CKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed