SCHEMBL20003048

SCHEMBL20003048

O=C(N1CCC(Sc2ccc(F)cc2)C1)N1CCO[C@H](CO)C1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 2/20 0.41
RORC P51449 2/20 0.39
CYP19A1 P11511 1/20 0.39
AKR1C3 P42330 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35
ALDH1A1 P00352 2/20 0.35
KMT2A Q03164 2/20 0.35
NR1H4 Q96RI1 1/20 0.35
CCR5 P51681 1/20 0.35
FKBP1A P62942 1/20 0.34
MAPT P10636 2/20 0.34
GAA P10253 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CCR3 P51677 3/20 0.34
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002992 1.00 PDK1 (0.41) PDK1RORCCYP19A1AKR1C3GRIN1
SCHEMBL20002879 0.77 NPC1 (0.44) GRIN1GRIN2BALDH1A1KMT2ACCR5
SCHEMBL20003024 0.76 NOTUM (0.44) AKR1C3GRIN1GRIN2BALDH1A1KMT2A
SCHEMBL20002297 0.76 NOTUM (0.47) RORCAKR1C3GRIN1GRIN2BKMT2A
SCHEMBL20002407 0.76 SMN1; SMN2 (0.41) AKR1C3GRIN1GRIN2BALDH1A1KMT2A
SCHEMBL20002936 0.76 CCR5 (0.46) AKR1C3GRIN1GRIN2BKMT2ACCR5
SCHEMBL28133029 0.74 PDK1 (0.62) PDK1RORCALOX5APFEN1KMT2A
SCHEMBL27785370 0.74 PDK1 (0.62) PDK1RORCALOX5APFEN1KMT2A
SCHEMBL28132263 0.74 PDK1 (0.62) PDK1RORCALOX5APFEN1KMT2A
SCHEMBL20002294 0.73 PTPN11 (0.36) RORCGRIN1GRIN2BKMT2ACCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed