SCHEMBL20002407

SCHEMBL20002407

CN1CCN(C(=O)N2CCC(Sc3ccc(F)cc3)C2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.41
HTT P42858 1/20 0.41
EPHX2 P34913 1/20 0.40
CCR5 P51681 1/20 0.39
KDM1A O60341 1/20 0.39
MAOB P27338 1/20 0.39
ALDH1A1 P00352 2/20 0.39
CYP2D6 P10635 1/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
RAB9A P51151 1/20 0.38
AKR1C3 P42330 1/20 0.38
KMT2A Q03164 1/20 0.38
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
MMP1 P03956 1/20 0.36
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36
MMP9 P14780 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002936 0.90 CCR5 (0.46) SMN1; SMN2CCR5AKR1C3KMT2AGRIN1
SCHEMBL20002879 0.88 NPC1 (0.44) SMN1; SMN2CCR5ALDH1A1NPC1LMNA
SCHEMBL20002297 0.85 NOTUM (0.47) CCR5NPC1RAB9AAKR1C3KMT2A
SCHEMBL20002294 0.83 PTPN11 (0.36) CCR5KMT2AGRIN1GRIN2BRIPK1
SCHEMBL20002612 0.82 RORC (0.36) CCR5NPC1RAB9AKMT2AGRIN1
SCHEMBL20003024 0.82 NOTUM (0.44) HTTEPHX2CCR5ALDH1A1NPC1
SCHEMBL9805869 0.77 POLB (0.50) SMN1; SMN2HTTKDM1AMAOBALDH1A1
SCHEMBL20002136 0.77 GPR119 (0.49) KMT2AMMP13
SCHEMBL20003227 0.77 KMT2A (0.38) SMN1; SMN2CCR5KDM1AMAOBKMT2A
SCHEMBL20003048 0.76 PDK1 (0.41) SMN1; SMN2CCR5ALDH1A1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed