SCHEMBL20002748

SCHEMBL20002748

COC1(C(=O)N2CCC([S+]([O-])c3ccc(F)cc3)C2)CCC(C)CC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RORC P51449 5/20 0.39
SMN1; SMN2 Q16637 4/20 0.36
RAB9A P51151 4/20 0.35
NPC1 O15118 3/20 0.35
ATM Q13315 1/20 0.34
HSD11B1 P28845 3/20 0.34
ALDH1A1 P00352 3/20 0.34
MAPT P10636 2/20 0.34
LMNA P02545 2/20 0.33
GAA P10253 2/20 0.33
HPGD P15428 1/20 0.33
PARP10 Q53GL7 1/20 0.33
KMT2A Q03164 1/20 0.33
PKM P14618 1/20 0.33
FAAH O00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002622 0.89 RORC (0.49) RORCSMN1; SMN2RAB9AHSD11B1ALDH1A1
SCHEMBL20003111 0.88 RORC (0.36) RORCSMN1; SMN2RAB9ANPC1ATM
SCHEMBL20002171 0.78 KMT2A (0.38) RORCSMN1; SMN2RAB9ANPC1ATM
SCHEMBL20003044 0.78 RORC (0.40) RORCSMN1; SMN2RAB9ANPC1ATM
SCHEMBL20002856 0.77 RORC (0.42) RORCSMN1; SMN2RAB9ANPC1ATM
SCHEMBL20002926 0.77 RORC (0.43) RORC
SCHEMBL20002561 0.77 RORC (0.50) RORCGAA
SCHEMBL20003110 0.77 RORC (0.41) RORC
SCHEMBL20003052 0.77 HSD11B1 (0.38) RORCSMN1; SMN2RAB9ANPC1ATM
SCHEMBL20002924 0.77 MAPK1 (0.34) RORCRAB9ANPC1ATMHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed