SCHEMBL20003097

SCHEMBL20003097

O=C(c1cccc(Cl)c1)N1CCC([S+]([O-])c2ccc(F)cc2)C1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 5/20 0.59
ALDH1A1 P00352 3/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
MGLL Q99685 2/20 0.48
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002981 0.81 KDM4E (0.55) HSD11B1ALDH1A1L3MBTL1SMN1; SMN2MEN1
SCHEMBL20002399 0.78 NAMPT (0.50) MGLL
SCHEMBL6211084 0.72 HSD11B1 (0.91) HSD11B1MGLLMEN1KMT2A
SCHEMBL20002698 0.72 HSD11B1 (0.47) HSD11B1ALDH1A1L3MBTL1SMN1; SMN2MEN1
SCHEMBL20002706 0.72 HSD11B1 (0.47) HSD11B1ALDH1A1L3MBTL1SMN1; SMN2MEN1
SCHEMBL20002958 0.71 NOTUM (0.48) HSD11B1ALDH1A1SMN1; SMN2KMT2A
SCHEMBL20002751 0.71 NOTUM (0.42) L3MBTL1
SCHEMBL20002969 0.71 NOTUM (0.45) HSD11B1ALDH1A1L3MBTL1SMN1; SMN2KMT2A
SCHEMBL20002167 0.71 KDM1A (0.40) ALDH1A1CYP2D6HTTSMN1; SMN2
SCHEMBL20002280 0.71 TACR1 (0.40) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed