SCHEMBL20003207

SCHEMBL20003207

CC(OC(I)(C(F)(F)F)C(F)(F)F)c1c(F)cccc1F

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.31
CES2 O00748 1/20 0.30
CES1 P23141 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002749 0.80 SCN1A (0.34) CES2CES1
SCHEMBL16886256 0.77 SCN1A (0.31)
SCHEMBL16892295 0.70 CES2 (0.36) CES2CES1
SCHEMBL9945893 0.65 ACHE (0.37) CES2CES1
SCHEMBL807556 0.64 CES2 (0.41) CES2CES1
SCHEMBL1604902 0.63 ALDH1A1 (0.38) CES2CES1
SCHEMBL28022516 0.63 CES2 (0.43) CES2CES1
SCHEMBL24498729 0.62 KCNK3 (0.40)
SCHEMBL4547921 0.62 P2RX7 (0.42) RORCCES2CES1
SCHEMBL1155196 0.61 DRD2 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed