SCHEMBL407809

SCHEMBL407809

NC(=O)C1(C(=O)Nc2ccc(F)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
MET P08581 10/20 0.49
LMNA P02545 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
AXL P30530 4/20 0.46
MERTK Q12866 4/20 0.46
GAA P10253 1/20 0.46
SPHK1 Q9NYA1 3/20 0.46
HDAC1 Q13547 1/20 0.46
RET P07949 1/20 0.46
KIT P10721 1/20 0.46
PDGFRA P16234 1/20 0.46
KDR P35968 1/20 0.46
FLT3 P36888 1/20 0.46
EGFR P00533 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL2458178 0.98 ALDH1A1 (0.55) ALDH1A1METLMNASMN1; SMN2AXL
Hydrochloric Acid SCHEMBL29453838 0.98 ALDH1A1 (0.55) ALDH1A1METLMNASMN1; SMN2AXL
SCHEMBL3856060 0.93 ALDH1A1 (0.53) ALDH1A1METLMNASMN1; SMN2AXL
Cadaverine Tartrate SCHEMBL29678843 0.90 ALDH1A1 (0.46) ALDH1A1METLMNASMN1; SMN2AXL
SCHEMBL12468984 0.89 ALDH1A1 (0.53) ALDH1A1METAXLMERTKGAA
SCHEMBL21299310 0.88 ALDH1A1 (0.55) ALDH1A1METLMNASMN1; SMN2AXL
SCHEMBL411823 0.85 ALDH1A1 (0.51) ALDH1A1METLMNASMN1; SMN2AXL
SCHEMBL19026688 0.85 MET (0.51) ALDH1A1METAXLMERTKGAA
SCHEMBL18256972 0.85 MET (0.54) ALDH1A1METAXLMERTKGAA
SCHEMBL105644 0.84 ALDH1A1 (0.48) ALDH1A1METAXLMERTKGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 188 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114040912-B Compounds for the treatment of kinase dependent disorders 埃克塞里艾克西斯公司 2024-10-25 CN claimed
CN-117919242-A Antitumor pharmaceutical composition 南昌弘益药业有限公司 2024-04-26 CN claimed
CN-116963734-A Crystalline salts of multiple tyrosine kinase inhibitors, process for their preparation and their use 米拉蒂治疗股份有限公司 2023-10-27 CN claimed
WO-2023193563-A1 CRYSTAL FORM A OF THIENOPYRIDINE COMPOUND, AND PREPARATION METHOD THEREFOR AND PHARMACEUTICAL COMPOSITION THEREOF 深圳海王医药科技研究院有限公司 2023-10-12 WO claimed
WO-2023155777-A1 N- [ (6-BROMOPYRIDIN-3-YL) METHYL] -2-METHOXYETHAN-1-AMINE SALTS AND PREPARATION THEREOF BEIGENE (SUZHOU) CO., LTD. (CN) 2023-08-24 WO claimed
US-11673897-B2 Compounds for the treatment of kinase-dependent disorders EXELIXIS, INC. (US) 2023-06-13 US claimed
US-20230167063-A1 Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms thereof for the treatment of cancer EXELIXIS, INC. 2023-06-01 US claimed
WO-2023056202-A2 COMPOSITIONS AND METHODS FOR ENHANCED PROTEIN PRODUCTION HDT BIO CORP. (US) 2023-04-06 WO claimed
CN-110386901-B Compound containing sulfonanilide pyrimidine structure and application thereof as antitumor drug 上海医药工业研究院 2022-11-25 CN claimed
WO-2022169248-A1 NOVEL COMPOUND AS PROTEIN KINASE INHIBITOR 주식회사 엘지화학 2022-08-11 WO claimed
EP-3329918-B1 C-MET MODULATORS AND METHODS OF USE EXELIXIS INC (US) 2022-05-25 EP claimed
CN-114401720-A Crystal form of polytyrosine kinase inhibitor, preparation method and application thereof 米拉蒂治疗股份有限公司 2022-04-26 CN claimed
CN-114040912-A Compounds for the treatment of kinase-dependent disorders 埃克塞里艾克西斯公司 2022-02-11 CN claimed
US-20210040076-A1 Compounds for the Treatment of Kinase-Dependent Disorders EXELIXIS, INC. 2021-02-11 US claimed
CN-105153028-B Compound as c-Met kinase inhibitor 南京爱德程医药科技有限公司 2019-03-26 CN claimed
CN-105683191-B Protein kinase inhibitor containing pyrrolopyridazine derivative 井标记生物 2019-03-26 CN claimed
WO-2009077874-A2 A PHARMACEUTICAL COMPOSITION FOR TREATING ESOPHAGEAL CANCER EISAI R & D MANAGEMENT CO., LTD. (US) 2009-06-25 WO claimed
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE, INC. 2007-01-04 US claimed
US-12503438-B2 Compounds for the treatment of kinase-dependent disorders EXELIXIS, INC. (US) 2025-12-23 US disclosed
US-20070054928-A1 c-Met modulators and methods of use EXELIXIS, INC. (US) 2007-03-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230167063-A1 Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms thereof for the treatment of cancer MDH1, MDH2, SLC25A11 ALDH1A1 819/4885MET 266/4885LMNA 3940/4885
US-20070054928-A1 c-Met modulators and methods of use FLT4, FLT1, MET ALDH1A1 2072/4885MET 3/4885LMNA 2924/4885
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling HGF, MET, FLT1 ALDH1A1 1649/4885MET 2/4885LMNA 4411/4885
US-20210040076-A1 Compounds for the Treatment of Kinase-Dependent Disorders ERBB2, MAP3K6, MAP3K1 ALDH1A1 3310/4885MET 154/4885LMNA 2013/4885
US-12503438-B2 Compounds for the treatment of kinase-dependent disorders ERBB2, ERBB3, PTK2B ALDH1A1 3579/4885MET 105/4885LMNA 2516/4885
US-11673897-B2 Compounds for the treatment of kinase-dependent disorders ERBB2, MAP3K6, PRKCH ALDH1A1 3263/4885MET 117/4885LMNA 1522/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.