SCHEMBL20005916

SCHEMBL20005916

c1ccc(CCC2CC3(C2)OCCO3)cc1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.40
MAOB P27338 3/20 0.40
KDM1A O60341 2/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
CTSC P53634 1/20 0.40
TAAR1 Q96RJ0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25415116 0.83 MAOA (0.44) MAOAMAOBSLC6A2SLC6A4SLC6A3
SCHEMBL7276325 0.75 KDM1A (0.46) MAOAMAOBKDM1ATAAR1
SCHEMBL582586 0.75 TSHR (0.44) CTSLCTSBCTSKTAAR1
SCHEMBL23809773 0.73 CARM1 (0.45) MAOAMAOBCTSLCTSBCTSS
SCHEMBL1609623 0.72 MAOA (0.58) MAOAMAOBCTSLCTSBCTSS
SCHEMBL15295395 0.72 MAOA (0.50) MAOAMAOBKDM1ASLC6A2SLC6A4
SCHEMBL25412651 0.71 MAOA (0.40) MAOAMAOBCTSLCTSBCTSS
SCHEMBL16572196 0.71 TAAR1 (0.49) MAOAMAOBSLC6A2SLC6A4SLC6A3
SCHEMBL16985344 0.70 CTSL (0.45) CTSLCTSBCTSSCTSKCTSC
SCHEMBL7616968 0.69 OPRM1 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2940019-B1 SUBSTITUTED SPIROPYRIDO[1,2-a]PYRAZINE DERIVATIVE AND MEDICINAL USE THEREOF AS HIV INTEGRASE INHIBITOR JAPAN TOBACCO INC (JP) 2018-03-28 EP disclosed