SCHEMBL7276325

SCHEMBL7276325

c1ccc(CCC2(CCc3ccccc3)OCCO2)cc1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.46
MAOA P21397 2/20 0.46
MAOB P27338 2/20 0.46
HMOX1 P09601 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
ALOX12 P18054 1/20 0.41
CASP1 P29466 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 2/20 0.39
CYP2A6 P11509 1/20 0.39
HTR2A P28223 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13536896 0.88 TDP1 (0.44) KDM1AMAOAMAOBHMOX1ALDH1A1
SCHEMBL13536901 0.85 KCNH2 (0.43) HTR2ASMN1; SMN2
SCHEMBL13536900 0.81 RAB9A (0.44) KDM1AMAOAMAOBTDP1SMN1; SMN2
SCHEMBL13536898 0.80 CYP1A2 (0.36) KDM1AMAOAMAOB
SCHEMBL1775344 0.80 HMOX1 (0.47) KDM1AMAOAMAOBHMOX1
SCHEMBL14130984 0.79 GAA (0.41) KDM1AMAOAMAOBALDH1A1HPGD
SCHEMBL15593870 0.77 TDP1 (0.41) MAOATDP1
SCHEMBL14779625 0.77 MAOA (0.46) KDM1AMAOAMAOB
SCHEMBL7269135 0.76 KDM1A (0.43) KDM1AMAOAMAOBALDH1A1HPGD
SCHEMBL20005916 0.75 MAOA (0.40) KDM1AMAOAMAOBTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed