SCHEMBL20007310

SCHEMBL20007310

N#Cc1ccc(S(=O)(=O)N2CCC(O)(CO)C2)nc1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 17/20 0.49
TRPM8 Q7Z2W7 1/20 0.42
CYP3A4 P08684 2/20 0.38
KCNH2 Q12809 2/20 0.38
CCR6 P51684 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20007811 0.88 TRPV4 (0.41) TRPV4TRPM8CYP3A4KCNH2
SCHEMBL23613990 0.83 TRPV4 (0.41) TRPV4
SCHEMBL20007693 0.83 TRPV4 (0.41) TRPV4
SCHEMBL20007244 0.79 TRPV4 (0.46) TRPV4CCR6
SCHEMBL23613847 0.77 TRPV4 (0.57) TRPV4TRPM8
SCHEMBL23176371 0.76 TRPV4 (0.55) TRPV4TRPM8
SCHEMBL20003513 0.76 TRPV4 (0.61) TRPV4TRPM8
SCHEMBL23614016 0.76 TRPV4 (0.55) TRPV4TRPM8
SCHEMBL20003515 0.76 TRPV4 (0.52) TRPV4TRPM8
SCHEMBL20003510 0.76 TRPV4 (0.61) TRPV4TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018055524-A1 TRPV4 ANTAGONISTS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2018-03-29 WO disclosed