SCHEMBL20008279

SCHEMBL20008279

C=Cc1cccc(CCC=N)c1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
ALDH1A1 P00352 2/20 0.37
TSHR P16473 1/20 0.37
PLAU P00749 1/20 0.35
FAAH O00519 1/20 0.35
OPRM1 P35372 2/20 0.33
OPRD1 P41143 2/20 0.33
OPRK1 P41145 2/20 0.33
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
CYP2D6 P10635 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
POLB P06746 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3674435 0.85 TP53 (0.45) TP53TDP1ALDH1A1TSHRPLAU
SCHEMBL29375309 0.84 TP53 (0.52) TP53TDP1ALDH1A1TSHRFAAH
SCHEMBL595016 0.84 TP53 (0.52) TP53TDP1ALDH1A1TSHRFAAH
SCHEMBL1645656 0.82 TP53 (0.50) TP53TDP1ALDH1A1TSHRPLAU
SCHEMBL29619562 0.82 TP53 (0.50) TP53TDP1ALDH1A1TSHRPLAU
SCHEMBL1646925 0.80 TP53 (0.48) TP53TDP1ALDH1A1TSHRFAAH
SCHEMBL29619625 0.80 TP53 (0.48) TP53TDP1ALDH1A1TSHRFAAH
SCHEMBL595251 0.79 TP53 (0.47) TP53TDP1ALDH1A1TSHRFAAH
SCHEMBL10616284 0.79 ALDH1A1 (0.52) TP53TDP1ALDH1A1TSHRFAAH
SCHEMBL3679531 0.78 TDP1 (0.42) TP53TDP1ALDH1A1TSHRFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed