SCHEMBL20008359

SCHEMBL20008359

Cc1ccc(C)c(-c2cnc(C)c(N3CCCCC3)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.42
SIGMAR1 Q99720 1/20 0.39
MAPT P10636 7/20 0.38
ALDH1A1 P00352 1/20 0.38
MCOLN3 Q8TDD5 1/20 0.38
LMNA P02545 5/20 0.38
KDM4E B2RXH2 2/20 0.38
HTT P42858 2/20 0.38
NPC1 O15118 1/20 0.38
PKM P14618 1/20 0.38
RAB9A P51151 1/20 0.38
TP53 P04637 4/20 0.37
S1PR2 O95136 1/20 0.36
STAT6 P42226 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HIF1A Q16665 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20009443 0.85 RAF1 (0.37) CNR2
SCHEMBL20008486 0.84 CNR2 (0.45) CNR2ALDH1A1HTTSMN1; SMN2POLB
SCHEMBL20008341 0.84 RAF1 (0.38)
SCHEMBL20050071 0.75 CYP2A6 (0.47) MAPTALDH1A1KDM4ERAB9ASMN1; SMN2
SCHEMBL20008475 0.74 RAF1 (0.39)
SCHEMBL20008237 0.73 HRH4 (0.47) CNR2
SCHEMBL20008313 0.73 ROCK2 (0.41) CNR2MAPTALDH1A1MEN1KMT2A
SCHEMBL16727174 0.71 SLC18A3 (0.55) MAPTALDH1A1MCOLN3LMNAHTT
SCHEMBL20008778 0.70 RAF1 (0.37)
SCHEMBL1442527 0.70 CNR2 (0.43) CNR2MAPTALDH1A1KDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed