SCHEMBL20008486

SCHEMBL20008486

Cc1cnc(C)c(-c2cnc(C)c(N3CCCCC3)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.45
PDE10A Q9Y233 1/20 0.36
OPRK1 P41145 2/20 0.36
ROCK2 O75116 4/20 0.35
ROCK1 Q13464 4/20 0.35
CDC42BPB Q9Y5S2 4/20 0.35
FEN1 P39748 1/20 0.34
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
NCF1 P14598 1/20 0.33
VRK1 Q99986 1/20 0.33
RAF1 P04049 1/20 0.33
BRAF P15056 1/20 0.33
KMO O15229 2/20 0.33
ABL1 P00519 1/20 0.33
POLB P06746 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20008359 0.84 CNR2 (0.42) CNR2ALDH1A1HTTPOLBSMN1; SMN2
SCHEMBL20008469 0.83 CNR2 (0.38) CNR2PDE10AROCK2ROCK1CDC42BPB
SCHEMBL20008475 0.83 RAF1 (0.39) ROCK2ROCK1CDC42BPBRAF1BRAF
SCHEMBL20008296 0.79 SMARCA2 (0.40) CNR2PDE10AOPRK1RAF1BRAF
SCHEMBL20008328 0.79 CNR2 (0.48) CNR2ALDH1A1GAARAF1BRAF
SCHEMBL20009443 0.75 RAF1 (0.37) CNR2ROCK2ROCK1CDC42BPBRAF1
SCHEMBL20008381 0.75 RAF1 (0.45) RAF1BRAFGRIN1GRIN2B
SCHEMBL20008472 0.74 RAF1 (0.38) VRK1RAF1BRAF
SCHEMBL20008341 0.73 RAF1 (0.38) ROCK2ROCK1CDC42BPBRAF1BRAF
SCHEMBL20008216 0.73 RAF1 (0.47) ROCK2ROCK1CDC42BPBRAF1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed