SCHEMBL20008586

SCHEMBL20008586

Fc1ncc(Br)cc1N1CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.39
ALDH1A1 P00352 4/20 0.38
HTT P42858 2/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 5/20 0.36
PKM P14618 1/20 0.36
LMNA P02545 1/20 0.36
PRNP P04156 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
PPARG P37231 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
NR2E3 Q9Y5X4 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
HRH3 Q9Y5N1 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30811846 0.98 MAPT (0.37) MAPK1ALDH1A1HTTGAAMAPT
SCHEMBL31728274 0.95 CHRNB2 (0.37) MAPK1ALDH1A1HTTGAAMAPT
SCHEMBL31728438 0.84 ALDH1A1 (0.40) MAPK1ALDH1A1MAPTTSHRNPC1
SCHEMBL29360875 0.83 CCR5 (0.43) MAPK1ALDH1A1GAAMAPTLMNA
SCHEMBL16121167 0.83 CCR5 (0.43) MAPK1ALDH1A1GAAMAPTLMNA
SCHEMBL31128265 0.79 L3MBTL1 (0.39) ALDH1A1HTTGAAMAPTLMNA
SCHEMBL26917123 0.79 HTT (0.47) MAPK1ALDH1A1HTTGAAMAPT
SCHEMBL29858551 0.79 HTT (0.47) MAPK1ALDH1A1HTTGAAMAPT
SCHEMBL31728501 0.78 PDE10A (0.34) OPRK1
SCHEMBL31727997 0.77 CNR2 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed