SCHEMBL2001196

SCHEMBL2001196

Cc1n[nH]c(C)c1C(c1ccc(-c2ccc(F)cc2)cc1)N1CCN(C)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.43
SLC1A2 P43004 1/20 0.40
MAPT P10636 3/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CHRM2 P08172 2/20 0.39
ADRA2A P08913 2/20 0.39
CHRM1 P11229 2/20 0.39
DRD1 P21728 2/20 0.39
DRD3 P35462 2/20 0.39
SLC6A3 Q01959 2/20 0.39
KCNH2 Q12809 2/20 0.39
CYP2D6 P10635 2/20 0.39
LMNA P02545 2/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
CHRM3 P20309 1/20 0.39
ADRA1D P25100 1/20 0.39
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1999561 0.88 LMNA (0.46) ACHEMAPTHTTNPSR1CHRM2
SCHEMBL5207006 0.85 CYP2D6 (0.44) ACHESLC1A2MAPTHTTNPSR1
SCHEMBL1999534 0.81 P4HB (0.35) MAPTKCNH2LMNAGAAP4HB
SCHEMBL1997982 0.78 ACHE (0.43) ACHESLC1A2MAPTHTTNPSR1
Hydrochloric Acid SCHEMBL3321146 0.76 RPS6KB1 (0.43) MAPTNPSR1DRD3LMNAGAA
Hydrochloric Acid SCHEMBL3327830 0.76 MAPT (0.47) ACHEMAPTKCNH2LMNAGAA
SCHEMBL27982331 0.75 RPS6KB1 (0.43) ACHEMAPTNPSR1LMNAGAA
SCHEMBL7395502 0.75 CYP2D6 (0.66) ACHESLC1A2MAPTCHRM2ADRA2A
Hydrochloric Acid SCHEMBL3327180 0.74 RPS6KB1 (0.42) ACHEMAPTNPSR1DRD3LMNA
SCHEMBL1994268 0.72 ACHE (0.45) ACHESLC1A2HTTCHRM2ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960413-B2 Pyrazole compounds MERCK PATENT GMBH (DE) 2011-06-14 US disclosed
US-20060276650-A1 Pyrazole compounds MERCK PATENT GMBH (DE) 2006-12-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060276650-A1 Pyrazole compounds HTR1D, HTR1A, HTR3A ACHE 1185/4885SLC1A2 356/4885MAPT 2121/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.