SCHEMBL200194

SCHEMBL200194

O=C(O)C(O)c1ccsc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.52
MAPK1 P28482 1/20 0.52
ALOX5 P09917 1/20 0.49
LCK P06239 1/20 0.45
FYN P06241 1/20 0.45
DAO P14920 1/20 0.45
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
SLC1A3 P43003 2/20 0.38
SLC1A2 P43004 2/20 0.38
SLC1A1 P43005 2/20 0.38
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
BLM P54132 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9329422 1.00 LMNA (0.52) LMNAMAPK1ALOX5LCKFYN
SCHEMBL11520740 0.81 ALOX5 (0.47) LMNAMAPK1ALOX5LCKFYN
SCHEMBL10759383 0.81 ALOX5 (0.56) ALOX5LCKFYNDAOCES2
SCHEMBL14416057 0.81 ALOX5 (0.51) LMNAMAPK1ALOX5LCKFYN
SCHEMBL18734632 0.80 CYP2D6 (0.50) LMNAMAPK1ALOX5LCKFYN
SCHEMBL162736 0.80 SRC (0.50) LMNAMAPK1ALOX5LCKFYN
SCHEMBL14671259 0.79 ALOX5 (0.42) LMNAMAPK1ALOX5LCKFYN
SCHEMBL18169428 0.79 ALOX5 (0.42) LMNAMAPK1ALOX5LCKFYN
SCHEMBL6775406 0.79 CES2 (0.63) LMNAMAPK1ALOX5LCKFYN
Hydrochloric Acid SCHEMBL11244144 0.78 SRC (0.48) ALOX5LCKFYNDAOCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 111 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230277491-A1 PHARMACEUTICAL COMBINATION COMPRISING GLYCOLIC ACID AND L-ALANINE PAN MONTOJO FRANCISCO (DE) 2023-09-07 US disclosed
EP-4188358-A2 PHARMACEUTICAL COMBINATION COMPRISING GLYCOLIC ACID AND L-ALANINE OR PYRUVATE Pan-Montojo, Francisco (DE) 2023-06-07 EP disclosed
US-20220354808-A1 GLYCOLIC ACID PROTECTS AGAINST ISCHEMIC INSULTS PAN MONTOJO FRANCISCO (DE) 2022-11-10 US disclosed
US-11426372-B2 Glycolic acid protects against ischemic insults PAN MONTOJO FRANCISCO (DE) 2022-08-30 US disclosed
WO-2022023545-A2 PHARMACEUTICAL COMBINATION COMPRISING GLYCOLIC ACID AND L-ALANINE PAN MONTOJO FRANCISCO (DE) 2022-02-03 WO disclosed
EP-3377055-B1 GLYCOLIC ACID PROTECTS AGAINST ISCHEMIC INSULTS PAN MONTOJO FRANCISCO (DE) 2021-10-13 EP disclosed
US-20180325849-A1 GLYCOLIC ACID PROTECTS AGAINST ISCHEMIC INSULTS PAN MONTOJO FRANCISCO (DE) 2018-11-15 US disclosed
EP-3377055-A1 GLYCOLIC ACID PROTECTS AGAINST ISCHEMIC INSULTS Pan-Montojo, Francisco (DE) 2018-09-26 EP disclosed
US-9828594-B2 Nitrilases, nucleic acids encoding them and methods for making and using them BASF ENZYMES LLC (US) 2017-11-28 US disclosed
US-20160355801-A1 NITRILASES, NUCLEIC ACIDS ENCODING THEM AND METHODS FOR MAKING AND USING THEM VERENIUM CORPORATION 2016-12-08 US disclosed
EP-0424021-B1 Antimuscarinic bronchodilators PFIZER LTD (GB) 1994-03-02 EP disclosed
US-5171744-A Antimuscarinic bronchodilators PFIZER INC. (US) 1992-12-15 US disclosed
US-5089490-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-18 US disclosed
EP-0424021-A1 Antimuscarinic bronchodilators Pfizer Limited (GB) 1991-04-24 EP disclosed
US-4758556-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1988-07-19 US disclosed
US-4297489-A CEPHALOSPORINS BRISTOL-MYERS COMPANY (US) 1981-10-27 US disclosed
US-4278793-A ANTIBIOTICS, BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1981-07-14 US disclosed
US-4172196-A CEPHALOSPORINS BRISTOL-MYERS COMPANY (US) 1979-10-23 US disclosed
US-4112228-A BACTERICIDES BRISTOL-MYERS COMPANY (US) 1978-09-05 US disclosed
US-3985738-A ANTIBACTERIAL AGENTS BRISTOL-MYERS COMPANY (US) 1976-10-12 US disclosed