SCHEMBL15468467

SCHEMBL15468467

Sc1ccncc1-c1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.44
RPS6KA3 P51812 2/20 0.42
GCGR P47871 2/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PKM P14618 1/20 0.41
HPGD P15428 1/20 0.41
MAPK14 Q16539 1/20 0.41
PTGS2 P35354 1/20 0.40
LIMK1 P53667 1/20 0.40
MAPT P10636 1/20 0.40
KDR P35968 1/20 0.40
TDO2 P48775 1/20 0.39
CDC25B P30305 1/20 0.38
CSNK2A1 P68400 1/20 0.38
HIPK2 Q9H2X6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15468461 0.83 LMNA (0.46) SLC22A12RPS6KA3MAPK14MAPTKDR
SCHEMBL28279885 0.81 RPS6KA3 (0.63) SLC22A12RPS6KA3GCGRNPC1RAB9A
SCHEMBL20020060 0.80 RPS6KA3 (0.68) SLC22A12RPS6KA3
SCHEMBL20020113 0.80 SLC22A12 (0.44) SLC22A12RPS6KA3GCGRNPC1RAB9A
SCHEMBL24810003 0.76 SLC22A12 (0.44) SLC22A12RPS6KA3GCGRNPC1RAB9A
SCHEMBL28109293 0.76 CYP11B1 (0.50) SLC22A12RPS6KA3GCGRMAPK14PTGS2
SCHEMBL15468459 0.76 RPS6KA3 (0.39) SLC22A12RPS6KA3SMN1; SMN2KDM4EMAPT
SCHEMBL16938695 0.76 MAPT (0.55) SLC22A12RPS6KA3NPC1RAB9ASMN1; SMN2
SCHEMBL30851299 0.73 SLC22A12 (0.42) SLC22A12RPS6KA3GCGRNPC1RAB9A
SCHEMBL30851377 0.73 CYP11B2 (0.54) SLC22A12RPS6KA3GCGRNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2975025-A1 THIOACETATE COMPOUNDS, COMPOSITIONS AND METHODS OF USE Ardea Biosciences, Inc. (US) 2016-01-20 EP disclosed
EP-2712861-B1 Thioacetate compounds, compositions and methods of use ARDEA BIOSCIENCES INC (US) 2015-07-29 EP disclosed
EP-2585437-B1 THIOACETATE COMPOUNDS, COMPOSITIONS AND METHODS OF USE ARDEA BIOSCIENCES INC (US) 2014-02-12 EP disclosed