SCHEMBL20021165

SCHEMBL20021165

Cc1cc2nc(CCc3ccccc3)ccc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.46
PLA2G2A P14555 1/20 0.44
LMNA P02545 1/20 0.41
DHODH Q02127 1/20 0.40
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
PTGDR2 Q9Y5Y4 5/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
MAOB P27338 1/20 0.38
ADORA1 P30542 1/20 0.38
CYP19A1 P11511 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20021173 0.87 PLA2G2A (0.40) KDM4EPLA2G2ADHODHESR1ESR2
SCHEMBL3323941 0.86 KDM4E (0.51) KDM4ESMN1; SMN2LMNADHODHPTGDR2
SCHEMBL20021110 0.84 KDM4E (0.45) KDM4ESMN1; SMN2LMNADHODHPTGDR2
SCHEMBL3297610 0.82 KDM4E (0.54) KDM4ESMN1; SMN2LMNADHODHPTGDR2
SCHEMBL3303954 0.82 KDM4E (0.53) KDM4ESMN1; SMN2LMNADHODHPTGDR2
SCHEMBL20021122 0.81 KDM4E (0.52) KDM4ESMN1; SMN2LMNADHODHPTGDR2
SCHEMBL20021074 0.79 KDM4E (0.44) KDM4ESMN1; SMN2DHODHPTGDR2MEN1
SCHEMBL3321643 0.79 KDM4E (0.48) KDM4ESMN1; SMN2LMNADHODHPTGDR2
SCHEMBL3314187 0.79 KDM4E (0.50) KDM4ESMN1; SMN2LMNADHODHPTGDR2
SCHEMBL3331488 0.79 KDM4E (0.51) KDM4ESMN1; SMN2LMNADHODHPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588455-B1 2-QUINOLINYL-ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES INC (US) 2018-04-04 EP disclosed