SCHEMBL20021173

SCHEMBL20021173

CCc1c(C)cc2nc(CCc3ccccc3)ccc2c1-c1ccc(Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 1/20 0.40
KDM4E B2RXH2 2/20 0.38
ESR1 P03372 2/20 0.38
ESR2 Q92731 2/20 0.38
CYP19A1 P11511 1/20 0.36
DHODH Q02127 2/20 0.35
FABP3 P05413 1/20 0.35
FABP4 P15090 1/20 0.35
FABP5 Q01469 1/20 0.35
KCNH2 Q12809 1/20 0.35
CYP3A4 P08684 1/20 0.35
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35
TUBB4B P68371 1/20 0.35
TUBB3 Q13509 1/20 0.35
TUBB2A Q13885 1/20 0.35
TUBB8 Q3ZCM7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20021165 0.87 KDM4E (0.52) PLA2G2AKDM4EESR1ESR2CYP19A1
SCHEMBL27928087 0.80 POLB (0.45) KDM4EESR1ESR2FABP3FABP4
SCHEMBL3323941 0.76 KDM4E (0.51) KDM4EDHODHFABP3FABP4FABP5
SCHEMBL245474 0.76 PLA2G2A (0.38) PLA2G2AESR1ESR2CYP19A1DHODH
SCHEMBL15182627 0.75 PLA2G2A (0.41) PLA2G2AESR1ESR2CYP19A1DHODH
SCHEMBL244126 0.75 PSIP1 (0.45) PLA2G2AESR1ESR2CYP19A1DHODH
SCHEMBL27921801 0.73 GPR84 (0.41) KDM4EFABP3FABP4FABP5KCNH2
SCHEMBL3342040 0.71 NOS1 (0.34) KDM4EDHODH
SCHEMBL20021110 0.71 KDM4E (0.45) KDM4EDHODHALDH1A1
SCHEMBL20021083 0.70 KMT2A (0.51) KDM4EKCNH2CYP3A4ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588455-B1 2-QUINOLINYL-ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES INC (US) 2018-04-04 EP disclosed