SCHEMBL20022720

SCHEMBL20022720

O=C(C1CC1)N1CCN(Cn2sc3c(C(F)(F)F)cccc3c2=O)CC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HB P07237 1/20 0.65
TGM2 P21980 1/20 0.41
EPHX2 P34913 2/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 2/20 0.38
ALDH1A1 P00352 2/20 0.37
ALDH1A2 O94788 1/20 0.37
ALDH2 P05091 1/20 0.37
ALDH3A1 P30838 1/20 0.37
ALDH1A3 P47895 1/20 0.37
MTNR1B P49286 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
SLC9A1 P19634 1/20 0.36
CYP2C19 P33261 1/20 0.36
SOS1 Q07889 1/20 0.35
CNR1 P21554 3/20 0.35
BRD4 O60885 1/20 0.34
PARP1 P09874 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20022721 0.86 P4HB (0.69) P4HBTGM2KDM4EMTNR1BCNR1
SCHEMBL20022718 0.85 P4HB (0.70) P4HBTGM2POLBALDH1A1ALDH1A2
SCHEMBL17948274 0.79 P4HB (1.00) P4HBTGM2ALDH1A1
SCHEMBL20022697 0.75 P4HB (0.69) P4HBTGM2
SCHEMBL21996081 0.72 P4HB (0.73) P4HBTGM2KDM4EALDH1A1ALDH1A2
SCHEMBL17948305 0.71 P4HB (0.72) P4HBEPHX2KDM4EALDH1A1MTNR1B
SCHEMBL21996048 0.71 P4HB (0.72) P4HBTGM2KDM4EPOLBALDH1A1
SCHEMBL21996082 0.70 MIF (0.47) P4HBALDH1A1ALDH3A1
SCHEMBL22056076 0.68 P4HB (0.58) P4HBEPHX2ALDH1A1ALDH1A2ALDH2
SCHEMBL20028779 0.66 P4HB (0.43) P4HBCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180092908-A1 SMALL MOLECULE OXIDIZERS OF PDI AND THEIR USE THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2018-04-05 US disclosed
US-20180092908-A1 SMALL MOLECULE OXIDIZERS OF PDI AND THEIR USE THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2018-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180092908-A1 SMALL MOLECULE OXIDIZERS OF PDI AND THEIR USE PDIA5, PDIA4, PDIA6 P4HB 5/4885TGM2 2410/4885EPHX2 1192/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.