SCHEMBL20031269

SCHEMBL20031269

CCc1nc(CC(=O)O)c(C(F)(F)F)o1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
AGBL2 Q5U5Z8 2/20 0.39
KDM4E B2RXH2 1/20 0.35
NOTUM Q6P988 1/20 0.32
FBP1 P09467 1/20 0.31
AKR1B1 P15121 1/20 0.31
GABRR1 P24046 1/20 0.30
DGAT1 O75907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17859504 0.80 FBP1 (0.44) AGBL2KDM4ENOTUMFBP1GABRR1
SCHEMBL3641559 0.69 FBP1 (0.53) KDM4EFBP1
SCHEMBL23723955 0.65 AGBL2 (0.45) GAAAGBL2KDM4ENOTUMGABRR1
SCHEMBL4675656 0.61 KDM4E (0.51) GAAAGBL2KDM4EGABRR1
SCHEMBL29733309 0.60 CYP1A2 (0.46) AGBL2KDM4EAKR1B1GABRR1
SCHEMBL11553826 0.60 L3MBTL1 (0.42) GAAKDM4E
SCHEMBL18359190 0.59 GAA (0.42) GAAAGBL2KDM4EGABRR1
SCHEMBL597035 0.59 DDR1 (0.41) GAAKDM4EDGAT1
SCHEMBL13765709 0.59 KDM4E (0.57) GAAAGBL2KDM4EGABRR1
SCHEMBL8947745 0.58 GABRP (0.34) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018059314-A1 AZABICYCLE DERIVATIVES AND PREPARATION METHOD AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2018-04-05 WO disclosed