SCHEMBL20037029

SCHEMBL20037029

CC(=N)/C(NC(=O)COC(=O)Cc1cccc(N)c1)=C(/C)Nc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
HTT P42858 1/20 0.49
KLK7 P49862 1/20 0.45
L3MBTL1 Q9Y468 3/20 0.43
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
GAA P10253 1/20 0.40
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GLS O94925 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20037101 0.90 KLK7 (0.55) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037030 0.89 ALDH1A1 (0.50) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037237 0.89 ALDH1A1 (0.50) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037082 0.89 KLK7 (0.53) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037121 0.88 ALDH1A1 (0.52) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037202 0.87 KLK7 (0.54) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037149 0.85 LMNA (0.47) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037052 0.85 ALDH1A1 (0.54) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037176 0.82 KLK7 (0.42) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037302 0.82 KLK7 (0.45) ALDH1A1HTTKLK7L3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018065607-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2018-04-12 WO disclosed
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed