SCHEMBL20037030

SCHEMBL20037030

CC(=N)/C(NC(=O)COC(=O)Cc1cccc(C)c1)=C(/C)Nc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
HTT P42858 2/20 0.50
KLK7 P49862 1/20 0.46
RECQL P46063 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
MAPK1 P28482 1/20 0.41
GAA P10253 2/20 0.41
NPC1 O15118 2/20 0.40
POLB P06746 2/20 0.40
RAB9A P51151 2/20 0.40
TP53 P04637 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40
PSENEN Q9NZ42 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20037101 0.90 KLK7 (0.55) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037237 0.90 ALDH1A1 (0.50) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037029 0.89 ALDH1A1 (0.49) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037121 0.89 ALDH1A1 (0.52) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037202 0.88 KLK7 (0.54) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037149 0.86 LMNA (0.47) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037052 0.85 ALDH1A1 (0.54) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037082 0.83 KLK7 (0.53) ALDH1A1HTTKLK7RECQLL3MBTL1
SCHEMBL20037302 0.83 KLK7 (0.45) ALDH1A1HTTKLK7L3MBTL1KMT2A
SCHEMBL20037113 0.82 KLK7 (0.70) ALDH1A1KLK7L3MBTL1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018065607-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2018-04-12 WO disclosed
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed