SCHEMBL20037880

SCHEMBL20037880

CCCN(C(=O)CC)c1ccc(C)nc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.38
OPRM1 P35372 4/20 0.37
MAPT P10636 2/20 0.37
KMT2A Q03164 1/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GPX4 P36969 1/20 0.35
RAB9A P51151 1/20 0.35
PAX8 Q06710 1/20 0.35
HCAR3 P49019 2/20 0.35
SIGMAR1 Q99720 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
MLYCD O95822 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2526618 0.76 MAPT (0.34) MAPTKMT2AHDAC1HDAC6
SCHEMBL20038496 0.74 CRHR1 (0.42) MAPTKMT2ANPC1RAB9AHCAR3
SCHEMBL18155441 0.73 TP53 (0.46) TP53OPRM1MAPTNPC1ALDH1A1
SCHEMBL2069920 0.73 TP53 (0.68) TP53OPRM1KMT2ANPC1ALDH1A1
SCHEMBL20038047 0.72 KMT2A (0.42) MAPTKMT2AHDAC1HDAC6ALDH1A1
SCHEMBL10893728 0.71 TRPM8 (0.55) TP53OPRM1MAPTNPC1ALDH1A1
SCHEMBL3634800 0.69 MLYCD (0.40) MAPTKMT2AHDAC1HDAC6NPC1
SCHEMBL11367960 0.68 NPC1 (0.64) TP53OPRM1NPC1ALDH1A1GPX4
SCHEMBL5429491 0.68 MLYCD (0.51) TP53MAPTKMT2AHDAC1HDAC6
SCHEMBL14337547 0.68 NOTUM (0.41) HDAC1HDAC6ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305785-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Teijin Pharma Limited (JP) 2018-04-11 EP disclosed