SCHEMBL20038036

SCHEMBL20038036

Cc1cc(OCCN2CCNCC2=O)cnc1I

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.34
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
SCN9A Q15858 1/20 0.33
HTR2C P28335 5/20 0.33
POLB P06746 1/20 0.32
KDM4E B2RXH2 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32
THRB P10828 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18291282 0.80 CHRNB2 (0.41) NPC1RAB9ASCN9AHTR2CCHRNB2
SCHEMBL20249280 0.74 NPC1 (0.38) PDK2NPC1RAB9ASCN9AKDM4E
SCHEMBL28830636 0.71 HRH2 (0.38) NPC1RAB9AHTR2CPOLBMEN1
SCHEMBL1596034 0.69 ALDH1A1 (0.36) SCN9AKDM4EMEN1KMT2A
Hydrochloric Acid SCHEMBL20745829 0.68 ALDH1A1 (0.36) SCN9AKDM4EMEN1KMT2A
SCHEMBL5337457 0.67 JAK2 (0.34) POLB
SCHEMBL20528090 0.65 MGLL (0.33) MEN1KMT2A
SCHEMBL15432724 0.65 MGLL (0.33) MEN1KMT2A
SCHEMBL20660200 0.64 DUT (0.39)
SCHEMBL1583740 0.64 MEN1 (0.35) NPC1RAB9AHTR2CPOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305785-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Teijin Pharma Limited (JP) 2018-04-11 EP disclosed