SCHEMBL20040174

SCHEMBL20040174

CNC(=N)c1ccc(C#C[Si](C)(C)C)cc1

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.32
APP P05067 1/20 0.32
ACACB O00763 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3941980 0.79 HDAC6 (0.50) GRM5ACACB
SCHEMBL28655847 0.77 MMP2 (0.34)
SCHEMBL1306384 0.76 GABRA1 (0.38) GRM5APP
SCHEMBL12934323 0.75 HDAC1 (0.38)
SCHEMBL1306505 0.73 APP (0.41) GRM5APP
SCHEMBL8049735 0.73 ALDH1A1 (0.43)
SCHEMBL9636621 0.72 HPGD (0.47) ACACB
SCHEMBL6036758 0.72 RARB (0.55) ACACB
SCHEMBL7262242 0.72 GABRA1 (0.31) GRM5
SCHEMBL168698 0.71 PTPN11 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2938599-B1 PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF BACTERIAL DISEASES JANSSEN SCIENCES IRELAND UC (IE) 2018-04-11 EP disclosed