SCHEMBL20041973

SCHEMBL20041973

COc1ccc(C2CN/C(=N\OCCOF)C2)cc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
PDE4A P27815 8/20 0.35
PDE4B Q07343 2/20 0.35
PDE4C Q08493 2/20 0.35
PDE4D Q08499 2/20 0.35
ADRA1A P35348 1/20 0.34
DRD2 P14416 1/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAP2K1 Q02750 1/20 0.32
MAOA P21397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16785342 0.86 TSHR (0.40) TSHRPDE4APDE4BPDE4CPDE4D
SCHEMBL19559484 0.86 TSHR (0.40) TSHRPDE4APDE4BPDE4CPDE4D
SCHEMBL20041975 0.81 TSHR (0.43) TSHRPDE4APDE4BPDE4CPDE4D
SCHEMBL19559451 0.81 TSHR (0.43) TSHRPDE4APDE4BPDE4CPDE4D
SCHEMBL19559581 0.76 TSHR (0.43) TSHRPDE4APDE4BPDE4CPDE4D
SCHEMBL19559443 0.72 TSHR (0.37) TSHRPDE4APDE4BPDE4CPDE4D
SCHEMBL20177592 0.70 ESRRG (0.34) TSHR
SCHEMBL20177943 0.70 HTR3A (0.36) TSHRADRA1ADRD2ALDH1A1SMN1; SMN2
SCHEMBL20177942 0.70 DRD2 (0.32) DRD2
SCHEMBL20177549 0.68 FPR1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305763-A1 DEUTERATED OR ISOTOPICALLY LABELED UREA DERIVATIVES OR PHARMACOLOGICALLY ACCEPTABLE SALTS THEREOF USEFUL AS FPRL-1 AGONISTS Kyorin Pharmaceutical Co., Ltd. (JP) 2018-04-11 EP disclosed