SCHEMBL20042663

SCHEMBL20042663

Cc1nc(O)c2c(n1)CN(C(=O)C(F)(F)F)C2

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 12/20 0.34
CYP1A2 P05177 1/20 0.32
CHRM4 P08173 1/20 0.32
ESR1 P03372 2/20 0.32
ESR2 Q92731 2/20 0.32
EP300 Q09472 1/20 0.32
CREBBP Q92793 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042664 0.84 P2RX7 (0.40) P2RX7CYP1A2CHRM4ESR1ESR2
SCHEMBL20042745 0.81 P2RX7 (0.33) P2RX7CYP1A2CHRM4EP300CREBBP
SCHEMBL20042855 0.77 P2RX7 (0.35) P2RX7CYP1A2CHRM4
SCHEMBL20042665 0.76 P2RX7 (0.32) P2RX7ESR1ESR2
SCHEMBL20078110 0.72 HSP90AA1 (0.52) ESR1ESR2
SCHEMBL19547099 0.71 P2RX7 (0.42) P2RX7
SCHEMBL13250465 0.68 PARP1 (0.47) ESR2
SCHEMBL30776241 0.68 PARP1 (0.47) ESR2
SCHEMBL30776218 0.68 ESR2 (0.45) ESR2
SCHEMBL20042726 0.67 PKM (0.45) P2RX7CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed