SCHEMBL20042745

SCHEMBL20042745

Cc1nc2c(c(N(C)C)n1)CN(C(=O)C(F)(F)F)C2

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 6/20 0.33
PDE10A Q9Y233 1/20 0.32
CYP1A2 P05177 1/20 0.30
CHRM4 P08173 1/20 0.30
EP300 Q09472 1/20 0.30
CREBBP Q92793 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042663 0.81 P2RX7 (0.34) P2RX7CYP1A2CHRM4EP300CREBBP
SCHEMBL20042664 0.80 P2RX7 (0.40) P2RX7CYP1A2CHRM4EP300CREBBP
SCHEMBL20042855 0.74 P2RX7 (0.35) P2RX7CYP1A2CHRM4
SCHEMBL20042665 0.73 P2RX7 (0.32) P2RX7
SCHEMBL20042749 0.70 PKM (0.43) P2RX7CYP1A2
SCHEMBL20078110 0.69 HSP90AA1 (0.52)
SCHEMBL20618233 0.63 NOTUM (0.36) P2RX7CYP1A2CHRM4CREBBP
SCHEMBL17106485 0.62 CYP1A2 (0.35) P2RX7CYP1A2CHRM4
SCHEMBL4266981 0.61 P2RX7 (0.45) P2RX7
SCHEMBL10028672 0.61 MAPT (0.43) CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed