SCHEMBL20042855

SCHEMBL20042855

Cc1nc2c(c(N3CC(F)C3)n1)CN(C(=O)C(F)(F)F)C2

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.35
CHRM4 P08173 11/20 0.34
CHRM2 P08172 2/20 0.34
CYP1A2 P05177 2/20 0.33
CHRM3 P20309 1/20 0.30
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042663 0.77 P2RX7 (0.34) P2RX7CHRM4CYP1A2
SCHEMBL20042664 0.76 P2RX7 (0.40) P2RX7CHRM4CYP1A2
SCHEMBL20042745 0.74 P2RX7 (0.33) P2RX7CHRM4CYP1A2
SCHEMBL20042793 0.71 SMN1; SMN2 (0.37) P2RX7CHRM4CYP1A2
SCHEMBL20042665 0.69 P2RX7 (0.32) P2RX7
SCHEMBL20042714 0.68 CHRM4 (0.43) CHRM4CYP1A2
SCHEMBL20042759 0.67 CHRM3 (0.35) CYP1A2CHRM3PDE4APDE4BPDE4C
SCHEMBL20042773 0.66 CHRM4 (0.52) CHRM4CHRM2CYP1A2
SCHEMBL20042806 0.66 CNR1 (0.47) CHRM4
SCHEMBL20042829 0.65 P2RX7 (0.41) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed