SCHEMBL20042669

SCHEMBL20042669

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)C1CC1c1ccccc1)C2

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.48
SIGMAR1 Q99720 3/20 0.47
HRH3 Q9Y5N1 11/20 0.46
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PREP P48147 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042660 0.79 CNR1 (0.39) MEN1ALDH1A1LMNATSHRKMT2A
SCHEMBL20042839 0.79 P2RX7 (0.45) MEN1ALDH1A1MAPTTSHRKMT2A
SCHEMBL20042729 0.78 HSD11B1 (0.43) LMNATSHR
SCHEMBL20042800 0.76 CNR1 (0.45) MEN1ALDH1A1LMNAMAPTTSHR
SCHEMBL20042806 0.76 CNR1 (0.47) MEN1ALDH1A1LMNAMAPTTSHR
SCHEMBL20042816 0.76 CNR1 (0.45) MEN1ALDH1A1LMNATSHRKMT2A
SCHEMBL20042748 0.74 NPC1 (0.49) ARMEN1ALDH1A1MAPTTSHR
SCHEMBL20042870 0.73 KDM4E (0.35) MEN1ALDH1A1LMNAMAPTTSHR
SCHEMBL20042776 0.73 P2RX7 (0.41) MEN1LMNATSHRKMT2A
SCHEMBL20042706 0.73 ALDH1A1 (0.43) ALDH1A1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed