SCHEMBL20042748

SCHEMBL20042748

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)CCc1ccccc1)C2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.46
GPBAR1 Q8TDU6 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
FKBP1A P62942 1/20 0.43
ALDH1A1 P00352 2/20 0.43
POLB P06746 2/20 0.43
NAAA Q02083 1/20 0.43
ME2 P23368 2/20 0.42
ME1 P48163 2/20 0.42
ME3 Q16798 2/20 0.42
KMT2A Q03164 2/20 0.41
GFER P55789 1/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
NPY5R Q15761 1/20 0.41
TSHR P16473 1/20 0.40
AR P10275 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042690 0.90 GFER (0.41) NPC1TDP1L3MBTL1GPBAR1ALDH1A1
SCHEMBL20042830 0.89 ME2 (0.43) NPC1TDP1GPBAR1FKBP1AALDH1A1
SCHEMBL20042688 0.89 C3AR1 (0.45) POLBKMT2AMEN1
SCHEMBL20042747 0.85 GRIN1 (0.39) GPBAR1FKBP1AKMT2A
SCHEMBL20042703 0.84 PTGDR2 (0.37)
SCHEMBL20042757 0.83 NPC1 (0.48) NPC1TDP1L3MBTL1GPBAR1HPGD
SCHEMBL20042730 0.83 NPC1 (0.48) NPC1TDP1L3MBTL1GPBAR1HPGD
SCHEMBL20042673 0.82 MAPK1 (0.38)
SCHEMBL20042714 0.79 CHRM4 (0.43) HPGDSMN1; SMN2ALDH1A1KMT2ATSHR
SCHEMBL20042654 0.78 HSD11B1 (0.41) SMN1; SMN2ALDH1A1KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed