SCHEMBL20042776

SCHEMBL20042776

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccnnc1)C2

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.41
PIK3CD O00329 1/20 0.37
GBA1 P04062 5/20 0.36
CNR1 P21554 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MTOR P42345 1/20 0.35
CFTR P13569 1/20 0.35
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
NR4A1 P22736 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HCAR2 Q8TDS4 1/20 0.34
GPR55 Q9Y2T6 2/20 0.34
ROCK2 O75116 1/20 0.34
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042832 0.88 CFTR (0.45) P2RX7SMN1; SMN2KDM4ECFTRLMNA
SCHEMBL20042755 0.86 GRM5 (0.43) P2RX7GBA1SMN1; SMN2KDM4ELMNA
SCHEMBL20042839 0.86 P2RX7 (0.45) P2RX7GBA1CNR1SMN1; SMN2KDM4E
SCHEMBL20042817 0.86 PKM (0.44) P2RX7GBA1KDM4ELMNAMEN1
SCHEMBL20042873 0.84 P2RX7 (0.38) P2RX7GBA1CNR1KDM4ECFTR
SCHEMBL20042872 0.84 P2RX7 (0.44) P2RX7GBA1CNR1SMN1; SMN2CFTR
SCHEMBL20042685 0.84 HTT (0.42) P2RX7GBA1SMN1; SMN2
SCHEMBL20042751 0.84 HSD17B10 (0.49) P2RX7GBA1SMN1; SMN2KDM4ELMNA
SCHEMBL20042743 0.83 P2RX7 (0.40) P2RX7GBA1CNR1SMN1; SMN2KDM4E
SCHEMBL20042912 0.83 PROKR1 (0.39) P2RX7PIK3CDGBA1CNR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed