SCHEMBL2004271

SCHEMBL2004271

CCOC(=O)c1cc(C(C)NS(=O)(=O)c2c(C)noc2C)ccc1-c1cc(F)ccc1OC

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 8/20 0.69
PGR P06401 8/20 0.69
MAPT P10636 4/20 0.39
GAA P10253 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
NR3C2 P08235 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004967 0.85 NR3C1 (0.76) NR3C1PGRMAPTGAAHSD17B10
SCHEMBL2006986 0.84 NR3C1 (0.72) NR3C1PGRMAPTGAAHSD17B10
SCHEMBL2011430 0.79 NR3C1 (0.78) NR3C1PGRMAPTGAAHSD17B10
SCHEMBL2011363 0.76 CETP (0.41) MAPTTSHRCCNT1CDK9LMNA
SCHEMBL2004253 0.67 NR3C1 (0.69) NR3C1PGRTP53
SCHEMBL2010050 0.64 NR3C1 (0.67) NR3C1PGRSMN1; SMN2POLB
SCHEMBL12161274 0.63 NR3C1 (0.49) NR3C1PGRMAPTTP53SMN1; SMN2
SCHEMBL2006930 0.62 NR3C1 (0.78) NR3C1PGRSMN1; SMN2ALDH1A1MEN1
SCHEMBL2532235 0.62 TSHR (0.54) MAPTGAATSHRSMN1; SMN2LMNA
SCHEMBL7008707 0.61 POLB (0.45) NR3C1MAPTTSHRNR3C2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960365-B2 Compounds with medicinal effects due to interaction with the glucocorticoid receptor N.V. ORGANON (NL) 2011-06-14 US disclosed
EP-1965785-A1 COMPOUNDS WITH MEDICINAL EFFECTS DUE TO INTERACTION WITH THE GLUCOCORTICOID RECEPTOR N.V. Organon (NL) 2008-09-10 EP disclosed
WO-2007071638-A1 COMPOUNDS WITH MEDICINAL EFFECTS DUE TO INTERACTION WITH THE GLUCOCORTICOID RECEPTOR N.V. ORGANON (NL) 2007-06-28 WO disclosed
US-20070149577-A1 Compounds with medicinal effects due to interaction with the glucocorticoid receptor N.V. ORGANON (NL) 2007-06-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070149577-A1 Compounds with medicinal effects due to interaction with the glucocorticoid receptor NR3C1, NR3C2, MC2R NR3C1 1/4885PGR 131/4885MAPT 2688/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.