SCHEMBL20042749

SCHEMBL20042749

Cc1nc2c(c(N(C)C)n1)CN(C(=O)c1cccc(Cl)c1)C2

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.43
P2RX7 Q99572 1/20 0.42
GRM5 P41594 4/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
ALDH1A1 P00352 5/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HSP90AA1 P07900 1/20 0.41
MAPT P10636 1/20 0.41
HTR1A P08908 1/20 0.41
HPGD P15428 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042726 0.85 PKM (0.45) PKMP2RX7GRM5CYP1A2CYP3A4
SCHEMBL20042862 0.84 HPGD (0.48) P2RX7ALDH1A1MEN1KMT2AMAPT
SCHEMBL20042920 0.83 GRM5 (0.41) P2RX7GRM5HSP90AA1HTR1A
SCHEMBL20042771 0.83 P2RX7 (0.47) PKMP2RX7GRM5CYP1A2CYP3A4
SCHEMBL20042737 0.77 P2RX7 (0.44) PKMP2RX7GRM5CYP1A2CYP3A4
SCHEMBL20042732 0.77 P2RX7 (0.44) PKMP2RX7GRM5CYP1A2CYP3A4
SCHEMBL20042739 0.77 P2RX7 (0.44) PKMP2RX7GRM5CYP1A2CYP3A4
SCHEMBL20042946 0.76 HPGD (0.46) P2RX7GRM5ALDH1A1L3MBTL1KDM4E
SCHEMBL20042734 0.74 P2RX7 (0.47) P2RX7GRM5ALDH1A1HPGD
SCHEMBL20042824 0.71 PROKR1 (0.40) KMT2AMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed