SCHEMBL20042734

SCHEMBL20042734

Cc1nc(Cl)c2c(n1)CN(C(=O)c1ccccc1)C2

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 6/20 0.47
MTHFD2 P13995 1/20 0.41
KIF11 P52732 1/20 0.41
HPGD P15428 1/20 0.41
GRM5 P41594 3/20 0.40
ACHE P22303 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
BLM P54132 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042744 0.86 MTHFD2 (0.44) P2RX7MTHFD2KIF11HPGDGRM5
SCHEMBL20042839 0.81 P2RX7 (0.45) P2RX7MTHFD2HPGDALDH1A1TSHR
SCHEMBL20042730 0.78 NPC1 (0.48) P2RX7HPGDALDH1A1TSHR
SCHEMBL20042726 0.77 PKM (0.45) P2RX7GRM5ALDH1A1
SCHEMBL20042749 0.74 PKM (0.43) P2RX7HPGDGRM5ALDH1A1
SCHEMBL25342146 0.74 MEN1 (0.44) P2RX7MTHFD2LMNATSHR
SCHEMBL20042664 0.74 P2RX7 (0.40) P2RX7
SCHEMBL20042751 0.74 HSD17B10 (0.49) P2RX7HPGDALDH1A1LMNA
SCHEMBL20042771 0.73 P2RX7 (0.47) P2RX7HPGDGRM5ALDH1A1LMNA
SCHEMBL11400880 0.71 PTGS1 (0.50) MTHFD2KIF11GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed