SCHEMBL20042763

SCHEMBL20042763

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)C1Cc3ccccc3C1)C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.39
TSHR P16473 2/20 0.39
LMNA P02545 2/20 0.39
NR4A1 P22736 1/20 0.39
GBA1 P04062 3/20 0.37
P2RX7 Q99572 1/20 0.36
PREP P48147 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KEAP1 Q14145 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
ALDH1A1 P00352 2/20 0.35
USP2 O75604 1/20 0.35
GAA P10253 1/20 0.35
CNR1 P21554 2/20 0.35
GPR55 Q9Y2T6 2/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
NPY5R Q15761 1/20 0.35
PDK1 Q15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042800 0.83 CNR1 (0.45) SMN1; SMN2TSHRLMNANR4A1GBA1
SCHEMBL20042806 0.83 CNR1 (0.47) SMN1; SMN2TSHRLMNANR4A1GBA1
SCHEMBL20042764 0.82 CNR1 (0.49) SMN1; SMN2TSHRLMNANR4A1GBA1
SCHEMBL20042660 0.81 CNR1 (0.39) SMN1; SMN2TSHRLMNANR4A1GBA1
SCHEMBL20042816 0.81 CNR1 (0.45) SMN1; SMN2TSHRLMNANR4A1GBA1
SCHEMBL20042793 0.81 SMN1; SMN2 (0.37) SMN1; SMN2TSHRLMNANR4A1GBA1
SCHEMBL20042669 0.80 AR (0.48) TSHRLMNAPREPMEN1KMT2A
SCHEMBL20042706 0.80 ALDH1A1 (0.43) SMN1; SMN2TSHRLMNANR4A1ALDH1A1
SCHEMBL20042839 0.79 P2RX7 (0.45) SMN1; SMN2TSHRGBA1P2RX7MEN1
SCHEMBL20042779 0.79 GPR55 (0.39) SMN1; SMN2TSHRLMNANR4A1GBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed