SCHEMBL20042650

SCHEMBL20042650

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)[C@@H](C)CC1CCCC1)C2

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
USP19 O94966 16/20 0.37
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
CYP1A2 P05177 1/20 0.34
CHRM4 P08173 1/20 0.34
NPY5R Q15761 1/20 0.34
CNR1 P21554 1/20 0.34
GPR55 Q9Y2T6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042651 0.82 CHRM4 (0.52) ADORA2AADORA1CYP1A2CHRM4NPY5R
SCHEMBL20042806 0.80 CNR1 (0.47) CHRM4CNR1GPR55
SCHEMBL20042654 0.80 HSD11B1 (0.41) ADORA2AADORA1CYP1A2CHRM4CNR1
SCHEMBL20042773 0.80 CHRM4 (0.52) ADORA2AADORA1CYP1A2CHRM4NPY5R
SCHEMBL20042764 0.79 CNR1 (0.49) CNR1GPR55
SCHEMBL20042834 0.78 CHRM4 (0.56) ADORA2AADORA1CYP1A2CHRM4CNR1
SCHEMBL20042714 0.76 CHRM4 (0.43) ADORA2AADORA1CYP1A2CHRM4CNR1
SCHEMBL20042816 0.75 CNR1 (0.45) CYP1A2CHRM4CNR1GPR55
SCHEMBL20042735 0.75 CNR2 (0.41) CHRM4CNR1GPR55
SCHEMBL20042706 0.74 ALDH1A1 (0.43) CHRM4CNR1GPR55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed