SCHEMBL20042784

SCHEMBL20042784

Cc1nc2c(c(N3CC(C)C3)n1)CN(C(=O)c1ccc(F)c(C#N)c1)C2

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.38
P2RX7 Q99572 1/20 0.38
FASN P49327 1/20 0.37
KDM1A O60341 9/20 0.36
PDK1 Q15118 3/20 0.36
PDK2 Q15119 3/20 0.36
ALDH1A1 P00352 1/20 0.35
LRRK2 Q5S007 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042783 0.93 GRM5 (0.38) GRM5P2RX7FASNKDM1AALDH1A1
SCHEMBL20042754 0.89 MEN1 (0.41) GRM5P2RX7FASNKDM1AALDH1A1
SCHEMBL20042696 0.81 KDM1A (0.45) GRM5P2RX7KDM1AALDH1A1
SCHEMBL20042903 0.79 MEN1 (0.42) P2RX7FASNALDH1A1
SCHEMBL20042666 0.77 KMT2A (0.46) GRM5P2RX7
SCHEMBL20042821 0.77 MEN1 (0.41) P2RX7FASNALDH1A1LRRK2
SCHEMBL20042698 0.76 MEN1 (0.43) P2RX7FASNALDH1A1LRRK2
SCHEMBL20042836 0.76 P2RX7 (0.43) P2RX7ALDH1A1
SCHEMBL20042733 0.75 MEN1 (0.41) P2RX7FASNALDH1A1
SCHEMBL20042667 0.75 TACR3 (0.46) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed