SCHEMBL20042836

SCHEMBL20042836

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccc(F)c(C)c1)C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.43
PDE2A O00408 3/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
GPR55 Q9Y2T6 1/20 0.39
GBA1 P04062 4/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TACR3 P29371 2/20 0.37
PIM1 P11309 1/20 0.36
TP53 P04637 2/20 0.35
HPGD P15428 2/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 3/20 0.35
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
THRB P10828 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042666 0.93 KMT2A (0.46) P2RX7PDE2ACNR1CNR2GPR55
SCHEMBL20042823 0.92 P2RX7 (0.45) P2RX7CNR1CNR2GPR55GBA1
SCHEMBL20042671 0.90 P2RX7 (0.45) P2RX7CNR1CNR2GPR55GBA1
SCHEMBL20042667 0.90 TACR3 (0.46) P2RX7PDE2ATACR3
SCHEMBL20042754 0.88 MEN1 (0.41) P2RX7MEN1KMT2AHPGDMAPT
SCHEMBL20042792 0.88 TACR3 (0.46) P2RX7PDE2ACNR1CNR2GPR55
SCHEMBL20042887 0.87 GPR6 (0.42) P2RX7CNR1CNR2GPR55GBA1
SCHEMBL20042685 0.87 HTT (0.42) P2RX7GBA1TACR3HTTSMN1; SMN2
SCHEMBL20042752 0.86 HPGD (0.47) P2RX7CNR1CNR2GPR55GBA1
SCHEMBL20042696 0.86 KDM1A (0.45) P2RX7MEN1KMT2AHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed