SCHEMBL20042666

SCHEMBL20042666

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccc(F)c(F)c1)C2

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
P2RX7 Q99572 1/20 0.43
TACR3 P29371 3/20 0.43
PDE2A O00408 3/20 0.39
HSD11B1 P28845 1/20 0.39
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
GABRA2 P47869 1/20 0.37
PGR P06401 1/20 0.36
GBA1 P04062 2/20 0.36
GRM5 P41594 2/20 0.36
KCNH2 Q12809 1/20 0.36
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042823 0.93 P2RX7 (0.45) KMT2AMEN1P2RX7TACR3HSD11B1
SCHEMBL20042836 0.93 P2RX7 (0.43) KMT2AMEN1P2RX7TACR3PDE2A
SCHEMBL20042792 0.91 TACR3 (0.46) KMT2AMEN1P2RX7TACR3PDE2A
SCHEMBL20042667 0.91 TACR3 (0.46) P2RX7TACR3PDE2AKCNH2
SCHEMBL20042696 0.89 KDM1A (0.45) KMT2AMEN1P2RX7GRM5
SCHEMBL20042754 0.89 MEN1 (0.41) KMT2AMEN1P2RX7GRM5
SCHEMBL20042882 0.89 P2RX7 (0.41) KMT2AMEN1P2RX7TACR3CNR1
SCHEMBL20042685 0.88 HTT (0.42) P2RX7TACR3HSD11B1GBA1GRM5
SCHEMBL20042752 0.87 HPGD (0.47) KMT2AMEN1P2RX7TACR3CNR1
SCHEMBL20042671 0.87 P2RX7 (0.45) KMT2AP2RX7CNR1CNR2GPR55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed