SCHEMBL20042868

SCHEMBL20042868

Cc1cc(Cl)cc(C(=O)N2Cc3nc(C)nc(N4CCC4)c3[C@H]2C)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.35
GRM5 P41594 1/20 0.35
TP53 P04637 2/20 0.34
POLB P06746 1/20 0.34
THRB P10828 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
LMNA P02545 2/20 0.33
TACR1 P25103 1/20 0.33
TACR2 P21452 1/20 0.33
TACR3 P29371 1/20 0.33
KCNH2 Q12809 1/20 0.33
HPGD P15428 1/20 0.32
FABP3 P05413 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
FABP4 P15090 1/20 0.32
FABP5 Q01469 1/20 0.32
KDM4E B2RXH2 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042876 0.90 TAS1R3 (0.40) P2RX7GRM5TP53THRBTDP1
SCHEMBL20042986 0.90 TAS1R3 (0.40) P2RX7GRM5TP53THRBTDP1
SCHEMBL20042853 0.88 GPR6 (0.34) P2RX7TP53THRBTDP1LMNA
SCHEMBL20042841 0.87 TACR2 (0.45) GRM5TP53THRBTDP1LMNA
SCHEMBL20042982 0.86 P2RX7 (0.46) P2RX7TP53POLBTHRBTDP1
SCHEMBL20042851 0.86 P2RX7 (0.46) P2RX7TP53POLBTHRBTDP1
SCHEMBL20042742 0.86 PROKR1 (0.35) P2RX7TP53POLBTHRBTDP1
SCHEMBL20043019 0.85 POLB (0.34) P2RX7GRM5TP53POLBTDP1
SCHEMBL20042852 0.83 TACR3 (0.47) P2RX7TACR1TACR2TACR3KCNH2
SCHEMBL20042883 0.83 GPR6 (0.39) P2RX7TP53THRBTDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed