SCHEMBL20042901

SCHEMBL20042901

Cc1nc2c(c(N3CCC3)n1)C(C)N(C(=O)N1Cc3ccccc3C1)C2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.38
HRH3 Q9Y5N1 4/20 0.38
NOTUM Q6P988 2/20 0.36
KDM4E B2RXH2 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RIPK1 Q13546 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KEAP1 Q14145 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTT P42858 1/20 0.34
NPY5R Q15761 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
GPR55 Q9Y2T6 1/20 0.34
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042971 0.89 NAMPT (0.37)
SCHEMBL20042913 0.84 PREP (0.37) KDM4ESMN1; SMN2MEN1KMT2AKEAP1
SCHEMBL31614760 0.79 SMN1; SMN2 (0.36) KDM4ESMN1; SMN2MEN1KMT2AHPGD
SCHEMBL20042786 0.77 LMNA (0.36) KDM4ESMN1; SMN2ALDH1A1
SCHEMBL20042958 0.76 TACR3 (0.42) KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL20042865 0.76 TACR3 (0.42) KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL20042851 0.76 P2RX7 (0.46) KCNH2SMN1; SMN2KMT2AALDH1A1CYP2C9
SCHEMBL20042982 0.76 P2RX7 (0.46) KCNH2SMN1; SMN2KMT2AALDH1A1CYP2C9
SCHEMBL20042990 0.76 CNR1 (0.37) KDM4ESMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL20042742 0.76 PROKR1 (0.35) KCNH2KDM4ESMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed