SCHEMBL2004404

SCHEMBL2004404

COc1ccc2c(c1)c(C(=O)c1nnc(-c3cnccn3)s1)cn2Cc1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.49
LMNA P02545 4/20 0.47
ALDH1A1 P00352 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.44
MAPT P10636 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
TERT O14746 1/20 0.41
PTGS2 P35354 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
PLA2G2A P14555 2/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004951 0.89 AHR (0.54) AHRLMNAALDH1A1SMN1; SMN2MAPT
SCHEMBL2003656 0.89 AHR (0.49) AHRLMNAALDH1A1SMN1; SMN2MAPT
SCHEMBL2005580 0.89 LMNA (0.47) AHRLMNAALDH1A1SMN1; SMN2MAPT
SCHEMBL2004829 0.87 AHR (0.50) AHRLMNAALDH1A1SMN1; SMN2MAPT
SCHEMBL2002890 0.87 AHR (0.49) AHRLMNAALDH1A1SMN1; SMN2MAPT
SCHEMBL2006518 0.86 LMNA (0.47) AHRLMNAALDH1A1SMN1; SMN2MAPT
SCHEMBL1998380 0.86 AHR (0.49) AHRLMNAALDH1A1SMN1; SMN2MAPT
SCHEMBL2012463 0.85 LMNA (0.56) AHRLMNAALDH1A1SMN1; SMN2MAPT
SCHEMBL2010072 0.84 LMNA (0.49) AHRLMNAALDH1A1SMN1; SMN2MAPT
SCHEMBL2006822 0.84 LMNA (0.47) AHRLMNAALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed